MCOPPB

CAS 1028969-49-4 MFCD128969494

化学结构图

1028969-49-4
SMILES: CC1(N2CCC(n3c([C@@H]4CCCNC4)nc4ccccc43)CC2)CCCCCCC1

化学属性

Mol. Weight408.6226
Appearance white to off-white solid powder
SolubilitySoluble in DMSO, not in water

别名和识别编码

Chemical NameMCOPPB
FormulaC26H40N4
Synonym MCOPPB
IUPAC Name(R)-1-(1-(1-methylcyclooctyl)piperidin-4-yl)-2-(piperidin-3-yl)-1H-benzo[d]imidazole
InChIKeyCYYNMPPFEJPBJD-OAQYLSRUSA-N
InChIInChI=1S/C26H40N4/c1-26(15-7-3-2-4-8-16-26)29-18-13-22(14-19-29)30-24-12-6-5-11-23(24)28-25(30)21-10-9-17-27-20-21/h5-6,11-12,21-22,27H,2-4,7-10,13-20H2,1H3/t21-/m1/s1
Canonical SMILESCC1(N2CCC(N3C([C@H]4CNCCC4)=NC5=CC=CC=C35)CC2)CCCCCCC1
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产品应用

  • MCOPPB is a drug which acts as a potent and selective agonist for the nociceptin receptor, with a pKi of 10.07 and much weaker activity at other opioid receptors. It has only moderate affinity for the mu opioid receptor, weak affinity for the kappa opioid receptor and negligible binding at the delta opioid receptor. In animal studies, MCOPPB produces potent anxiolytic effects, with no inhibition of memory or motor function, and only slight sedative side effects which do not appear until much higher doses than the effective anxiolytic dose range. (http://en.wikipedia.org/wiki/MCOPPB)

安全信息

Storage condition Dry, dark and at 0 - 4 C for short term (days to weeks) or -20 C for long term (months to years).

系列性分类

  1. Medical Research Areas
  2. Endocrinology & Hormones
  3. Opioid Receptor
  1. Medical Research Areas
  2. GPCR & G Protein
  3. Opioid Receptor
  1. Medical Research Areas
  2. Neuronal Signaling
  3. Opioid Receptor

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